BTK INHIBITOR
PCT/CN2015/081686
[WANG, Xuehai 王学海, WANG, Xuehai 王学海, WU, Chengde 吴成德, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, YANG, Jing 杨菁, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, YANG, Jing 杨菁, TANG, Jing 唐静, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, YANG, Jing 杨菁, TANG, Jing 唐静, ZHOU, Wen 周文, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, YANG, Jing 杨菁, TANG, Jing 唐静, ZHOU, Wen 周文, YU, Jing 于静, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, YANG, Jing 杨菁, TANG, Jing 唐静, ZHOU, Wen 周文, YU, Jing 于静, ZHANG, Yi 张毅, WANG, Xuehai 王学海, WU, Chengde 吴成德, XU, Yong 许勇, SHEN, Chunli 沈春莉, LI, Li'e 李莉娥, HU, Guoping 胡国平, YUE, Yang 乐洋, LI, Jian 黎健, GUO, Diliang 郭涤亮, SHI, Nengyang 施能扬, HUANG, Lu 黄璐, CHEN, Shuhui 陈曙辉, TU, Ronghua 涂荣华, YANG, Zhongwen 杨仲文, ZHANG, Xuwen 张绪文, XIAO, Qiang 肖强, TIAN, Hua 田华, YU, Yanping 余艳平, CHEN, Hailiang 陈海靓, SUN, Wenjie 孙文洁, HE, Zhenyu 何震宇, SHEN, Jie 沈洁, YANG, Jing 杨菁, TANG, Jing 唐静, ZHOU, Wen 周文, YU, Jing 于静, ZHANG, Yi 张毅, LIU, Quan 刘荃]
No.666 Gaoxin Road, Wuhan East Lake Hi-tech Development Zone 中国湖北省武汉市东湖高新技术开发区高新大道666号, Hubei 430075Wuhan, Hubei 430075;No.666 Gaoxin Road, Wuhan East Lake Hi-tech Development Zone 中国湖北省武汉市武汉东湖开发区高新大道666号, Hubei 430075Wuhan, Hubei 430075
Provided are a series of BTK inhibitors, and specifically disclosed are a compound, pharmaceutically acceptable salt thereof, tautomer thereof or pro-drug thereof represented by formula (I), (II), (III) or (IV).
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